Tislelizumab

Tislelizumab
Fab fragment of tislelizumab (green) binding the extracellular domain of PD-1 (pale pink). From PDB entry 7BXA
Monoclonal antibody
TypeWhole antibody
SourceHumanized
TargetPD-1
Clinical data
Trade namesTevimbra
Other namesBGB-A317, tislelizumab-jsgr
AHFS/Drugs.comMonograph
MedlinePlusa624026
License data
Pregnancy
category
Routes of
administration
Intravenous
Drug classAntineoplastic agent
ATC code
Legal status
Legal status
Identifiers
CAS Number
DrugBank
ChemSpider
  • none
UNII
KEGG

Tislelizumab, sold under the brand name Tevimbra among others, is an anti-cancer medication used for the treatment of various forms of cancer. It is a humanized monoclonal antibody directed against programmed death receptor-1.[4] It is being developed by BeOne Medicines.[7]

Tislelizumab was approved for medical use in China in December 2019,[8][9] in the European Union in September 2023,[5] in the United States in March 2024,[10][11] and in Australia in May 2024.[1]

  1. ^ a b c "Tevimbra (tislelizumab)". Therapeutic Goods Administration (TGA). 28 June 2024. Retrieved 7 July 2024.
  2. ^ "Tevimbra (Beigene Aus Pty Ltd)". Therapeutic Goods Administration (TGA). 1 July 2024. Retrieved 7 July 2024.
  3. ^ "Tevimbra tislelizumab 100 mg/10 mL concentrated injection vial (391176)". Therapeutic Goods Administration (TGA). 31 May 2024. Retrieved 27 December 2024.
  4. ^ a b "Tevimbra- tislelizumab injection, solution, concentrate". DailyMed. 16 March 2024. Archived from the original on 2 April 2024. Retrieved 2 April 2024.
  5. ^ a b "Tevimbra EPAR". European Medicines Agency (EMA). 4 October 2023. Archived from the original on 28 November 2023. Retrieved 5 October 2023.
  6. ^ "Tevimbra Product information". Union Register of medicinal products. 19 September 2023. Retrieved 1 October 2023.
  7. ^ Cite error: The named reference GP3 was invoked but never defined (see the help page).
  8. ^ Lee A, Keam SJ (April 2020). "Tislelizumab: First Approval". Drugs. 80 (6): 617–624. doi:10.1007/s40265-020-01286-z. PMID 32185681.
  9. ^ "BeiGene scores first China OK with PD-1 — to be manufactured by Boehringer Ingelheim". Endpoints News. 2 January 2020. Archived from the original on 2 July 2020. Retrieved 1 July 2020.
  10. ^ "Novel Drug Approvals for 2024". U.S. Food and Drug Administration (FDA). 29 April 2024. Archived from the original on 30 April 2024. Retrieved 30 April 2024.
  11. ^ New Drug Therapy Approvals 2024 (PDF). U.S. Food and Drug Administration (FDA) (Report). January 2025. Archived from the original on 21 January 2025. Retrieved 21 January 2025.